Valeant Pharmaceuticals Highlights Taribavirin Phase IIb End of Study Data Presentation at American Association for the Study of
November 03 2009 - 8:00AM
PR Newswire (US)
ALISO VIEJO, Calif., Nov. 3 /PRNewswire-FirstCall/ -- Valeant
Pharmaceuticals (NYSE:VRX) today announced that results from the
week-72 analysis for its Phase IIb dose-finding clinical trial for
taribavirin, a prodrug of ribavirin which is in development for the
treatment of chronic hepatitis C in conjunction with a pegylated
interferon, were presented at the American Association for the
Study of Liver Disease (AASLD) 60th Annual Meeting in Boston. It is
believed that taribavirin (TBV) may present an alternative therapy
to ribavirin (RBV) for the treatment of hepatitis C by delivering
similar efficacy to ribavirin but with significantly less anemia,
which is the main treatment-limiting toxicity associated with
ribavirin. The results were presented in an abstract entitled
"Sustained Virologic Response Results for Weight-Based Taribavirin
Versus Weight-Based Ribavirin, in Naïve Chronic Hepatitis C,
Genotype 1 Patients", with an oral presentation given by Fred
Poordad, M.D., Chief of Hepatology at the Center for Liver Disease
and Transplant, Cedars-Sinai Medical Center, Los Angeles, CA and
principal investigator in this study. "The final results of this
Phase IIb study are promising, and imply that comparable efficacy
can be achieved when compared to ribavirin," said Dr. Poordad. "As
is known for ribavirin, low doses are associated with a high
relapse rate and, except for the lowest dose with taribavirin,
relapse rates are also comparable to ribavirin. The safety of this
ribavirin analog is of particular relevance in that its use is
associated with significantly less anemia in an evolving era of
small molecule therapies, where anemia appears to be more
problematic." The company has previously reported results from this
Phase IIb trial exploring weight- based dosing of taribavirin at
20, 25 and 30mg/kg vs. weight-base dosed ribavirin 800-1400mg. The
study consisted of 48 weeks of treatment with a 24-week
post-treatment follow-up period. Consistent with previous reports,
the viral response data continued to show comparable reductions in
viral load for weight-based doses of taribavirin and ribavirin in a
difficult-to-treat population of subjects infected with hepatitis C
genotype 1 and end-of-study sustained virologic response rates were
again comparable across the treatment groups. Relapse rates were
identical for taribavirin 25mg/kg and weight-based doses of
ribavirin. Importantly, the statistically significantly lower
anemia rate for patients receiving taribavirin in the 20mg/kg and
25mg/kg arms versus the ribavirin control arm has been maintained
at a rate similar to the end-of- treatment (week 48) throughout.
Table: Efficacy/Safety (intent-to-treat) Phase IIb --------- TBV
TBV TBV RBV 20 mg/kg 25 mg/kg 30 mg/kg 800-1400mg n=67 n=70 n=68
n=70
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TW4 Undetectable(1) 11 (16.4%) 10 (14.3%) 11 (16.2%) 8 (11.4%)
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TW12 Undetectable(1) 28 (41.8%) 29 (41.4%) 17 (25.0%) 22 (31.4%)
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TW48 Undetectable(1) 30 (44.8%) 27 (38.6%) 23 (33.8%) 26 (37.1%)
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SVR Undetectable(1) 19 (28.4%) 19 (27.1%) 19 (27.9%) 19 (27.1%)
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Relapse Rate 10 (34.5%) 5 (20.8%) 3 (13.6%) 5 (20.8%)
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Anemia 48 weeks(2) 9 (13.4%)* 11 (15.7%)* 19 (27.9%) 23 (32.9%)
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(1) HCV RNA < 39 IU/mL (2) Anemia: hemoglobin < 10g/dL
*P=400,000 IU/mL and 82.1 kg mean weight. Week 72 efficacy and
safety results for the intention-to-treat (ITT) population are
shown in the table above. About Valeant Valeant Pharmaceuticals
International (NYSE:VRX) is a multinational specialty
pharmaceutical company that develops, manufactures and markets a
broad range of pharmaceutical products primarily in the areas of
neurology and dermatology. More information about Valeant can be
found at http://www.valeant.com/. FORWARD-LOOKING STATEMENTS This
press release may contain forward-looking statements, including,
but not limited to, statements regarding the potential for
taribavirin in the treatment of hepatitis C, and the continuing
role of ribavirin or taribavirin in the treatment of hepatitis C,
Forward-looking statements may be identified by the use of the
words "anticipates," "expects," "intends," "plans," "should,"
"could," "would," "may," "will," "believes," "estimates,"
"potential," or "continue" and variations or similar expressions.
These statements are based upon the current expectations and
beliefs of management and are subject to certain risks and
uncertainties that could cause actual results to differ materially
from those described in the forward-looking statements. These risks
and uncertainties include, but are not limited to, risks and
uncertainties discussed in the company's most recent annual or
quarterly report filed with the U.S. Securities and Exchange
Commission, which factors are incorporated herein by reference.
Readers are cautioned not to place undue reliance on any of these
forward-looking statements. Valeant undertakes no obligation to
update any of these forward-looking statements to reflect events or
circumstances after the date of this press release or to reflect
actual outcomes. Contact: Laurie W. Little, Valeant Pharmaceuticals
949-461-6002 (Logo:
http://www.newscom.com/cgi-bin/prnh/20081125/VALEANTLOGO)
http://www.newscom.com/cgi-bin/prnh/20081125/VALEANTLOGO
http://photoarchive.ap.org/ DATASOURCE: Valeant Pharmaceuticals
International CONTACT: Laurie W. Little of Valeant Pharmaceuticals,
+1-949-461-6002, Web Site: http://www.valeant.com/
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