Alchemia’s HyACT Technology Enhances the Killing of Cancer Stem Cell Populations in Breast and Colorectal Cancer
April 20 2010 - 9:38PM
Business Wire
Alchemia’s (ASX: ACL) subsidiary Alchemia Oncology today
presented two posters at the American Association of Cancer
Research (AACR) 101st Annual Meeting in Washington, DC. The data
demonstrates the ability of the Company’s HyACT tumour targeting
technology to dramatically enhance the killing of cancer stem
cells. These cells are highly resistant to treatment with
chemotherapeutic drugs and are believed to be responsible for
treatment failure and disease recurrence.
Two posters were presented today at the ‘Cancer Stem Cell
Therapeutics 2’ session from 2:00-5:00pm EDT in Exhibit Hall A-C
entitled,
Poster #4278: HA-Irinotecan targeting
of activated CD44 is an effective therapy for the eradication of
putative colon cancer stem cells
Poster #4293: Evaluation of activated
CD44 as a biological target in the eradication of breast cancer
stem cells
In new data presented today by Professor Tracey Brown,
Alchemia’s Vice President of Preclinical Research, the HyACT
formulation of doxorubicin (HA-Doxorubicin) has been shown to be up
to forty times more potent than doxorubicin alone in killing
putative breast cancer stem cells. Similarly, in human colorectal
cancer cells, HyACT formulations of the drug irinotecan
(HA-Irinotecan) showed up to a fifty fold increase in potency
against stem cell like populations.
Despite advances in the treatment of cancer with new
chemotherapeutic agents and targeted therapies, many patients
develop tumours that are resistant to treatment, resulting in
treatment failure. In recent years, attention has focused on the
role of a sub-population of cells, referred to as ‘cancer stem
cells’, which are highly resistant to treatment. One of the markers
used to define this difficult to eradicate cell population is CD44,
which is specifically targeted by Alchemia’s HyACT technology.
“In previous research we have clearly established that
reformulation of cancer drugs with HyACT enhances the ability of
that drug to kill cells expressing the receptor CD44,” said
Professor Tracey Brown. “It is increasingly accepted that cancer
stem cells from a majority of solid tumours express high levels of
activated CD44. Our research presented today confirms that
targeting of drugs to that receptor with HyACT may help to
eradicate this otherwise difficult to treat population of cells.
Indeed, it may explain the significant increases in efficacy that
we have seen in previously reported Phase 2 clinical studies of
HA-Irinotecan in colorectal cancer and preclinical data from models
of several different cancer types.”
“The role of cancer stem cells in the genesis and progression of
the disease is receiving intense scrutiny in the research and
clinical communities,” said Pete Smith, CEO of Alchemia. “These
data provide additional excitement around the technology as we
prepare to start the pivotal Phase III study of HA-Irinotecan in
colorectal cancer.”
The posters presented at today’s session at AACR are now
available to view on Alchemia’s website:
www.alchemia.com.au/irm/content/investor_presentations.html
About Alchemia Limited – www.alchemia.com.au
Alchemia is a drug discovery and development Company founded on
its chemistry expertise. The Company’s lead program is fondaparinux
(a generic version of GlaxoSmithKline’s Arixtra®, a synthetic
anticoagulant mainly used for the prevention of deep vein
thrombosis). The ANDA for generic fondaparinux was filed for
approval with the US FDA in March 2009. Fondaparinux is expected to
generate positive cash-flows for the company commencing in the
second half of calendar 2010. It is partnered with Dr Reddy’s
Laboratories Inc. for the U.S. market. Alchemia’s pipeline of
assets is built on two platform technologies: HyACT® (targeted
cancer delivery) and VAST® (drug discovery). The primary objective
of the HyACT® technology is to develop a new generation of
anti-cancer drugs which demonstrate better efficacy. The lead
product from the HyACT® platform is HA-Irinotecan for which a phase
III clinical trial in metastatic colorectal cancer will commence in
2010. In addition to HA-Irinotecan, Alchemia has successfully taken
two other anti-cancer products HA-Doxorubicin (doxorubicin and
hyaluronic acid) and HA-Fluorouracil (5-fluorouracil and hyaluronic
acid) into successful Phase I clinical testing and they continue to
development on five other HyACT® drugs.
About AACR
AACR is a professional society of more than 24,000 laboratory
and clinical scientists engaged in basic, translational, and
clinical cancer research in the United States and more than 60
other countries. Its annual meeting is attended by more than 15,000
scientists from around the world who share new and significant
discoveries in the cancer field.
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