Immunome Presents Compelling Preclinical Data Demonstrating Robust Anti-Tumor Activity for IM-1021
October 29 2024 - 8:00AM
Business Wire
- IM-1021 showed superior potency when compared to a competitor
in both mantle cell lymphoma and triple-negative breast cancer
preclinical models; IND submission expected in 1Q25
- HC74, Immunome’s proprietary TOP1 ADC payload, shows superior
potency, desirable ADME properties, and enhanced efficacy in
chemo-resistant cell lines when compared to deruxtecan
Immunome, Inc. (Nasdaq: IMNM), a biotechnology company focused
on developing first-in-class and best-in-class targeted cancer
therapies, recently presented promising preclinical data for
IM-1021 and the associated proprietary ADC payload HC74. The
results were presented in a poster entitled “Preclinical evaluation
of IM-1021, a ROR1-targeted antibody-drug conjugate with a novel
topoisomerase I linker payload” at the 36th EORTC-NCI-AACR
Symposium on Molecular Targets and Cancer Therapeutics in Barcelona
on October 24, 2024.
The poster included preclinical results for IM-1021 in both
liquid and solid tumors while also highlighting the enhanced ADME
properties of HC74:
- IM-1021 showed superior efficacy compared to zilovertamab
vedotin in both the Jeko-1 mantle cell lymphoma model and the
MDA-MB-468 triple negative breast cancer model. In the MDA-MB-468
study, 5 out of 8 animals achieved complete responses after three 5
mg/kg doses.
- HC74 demonstrated superior potency (IC50=5nM) compared to
deruxtecan (IC50=20nM) in a panel of 89 cancer cell lines.
- HC74 showed faster hepatocyte clearance, higher permeability,
and lower efflux than deruxtecan.
- When evaluated in doxorubicin-resistant and
vincristine-resistant cell lines, HC74 showed no reduction in
potency compared to the parental NCI-H69 cell line.
Immunome expects to submit an IND for the IM-1021 program to the
FDA in the first quarter of 2025.
“We believe that transformative ADCs require matching the target
with the right combination of antibody, linker, and payload. Based
on this data, we continue to believe that IM-1021 is a promising
preclinical candidate,” said Immunome’s Chief Scientific Officer
Jack Higgins, Ph.D. “HC74’s differentiated profile, including
substantial potency in chemo-resistant cell lines, provides
intriguing opportunities for clinical development. We look forward
to submitting the IM-1021 IND and starting clinical trials upon IND
clearance to further validate these findings.”
A copy of the poster is available in the “Events &
Presentations” portion of Immunome’s website.
About Immunome, Inc.
Immunome is a clinical-stage targeted oncology company committed
to developing first- and best-in-class targeted therapies designed
to improve outcomes for cancer patients. We are advancing an
innovative portfolio of therapeutics, drawing on leadership that
previously played key roles in the design, development, and
commercialization of cutting-edge targeted cancer therapies,
including antibody-drug conjugate therapies (ADCs.) In addition to
a portfolio of discovery-stage ADCs, our pipeline includes AL102, a
gamma secretase inhibitor which is currently in a Phase 3 trial for
treatment of desmoid tumors, as well as IM-1021, a ROR1 ADC, and
IM-3050, a FAP-targeted radioligand, both of which are the subject
of INDs expected to be submitted in the first quarter of 2025. For
more information, visit www.immunome.com.
Cautionary Statement Regarding Forward-Looking
Statements
Statements in this press release that are not purely historical
in nature are “forward-looking statements” within the meaning of
the Private Securities Litigation Reform Act of 1995. We use words
such as “expected,” “expects,” “believe,” “promising,” “look
forward” and similar expressions to identify these forward-looking
statements. These forward-looking statements include, but are not
limited to, Immunome’s expected timing for submission of an IND for
IM-1021 and IM-3050; Immunome’s ability to initiate clinical
studies for IM-1021; the potential benefits and drug profile of
IM-1021 and HC74; and other statements regarding management’s
intentions, plans, beliefs, expectations or forecasts for the
future. These forward-looking statements are based on Immunome’s
current expectations and involve assumptions that may never
materialize or may prove to be incorrect; consequently, actual
results may differ materially from those expressed or implied in
the statements due to a number of factors, including, but not
limited to, the risk that Immunome will not be able to realize the
benefits of its strategic transactions; the risk that regulatory
approvals for Immunome’s product candidates are not obtained, are
delayed or are subject to unanticipated conditions; the risk that
pre-clinical data may not be predictive of clinical data; the risk
that Immunome’s product candidates fail to achieve their intended
endpoints; and other risks and uncertainties indicated from time to
time described in Immunome’s Quarterly Report on Form 10-Q for the
quarter ended June 30, 2024, filed with the SEC on August 12, 2024,
and in Immunome’s other filings with the SEC. Except as required by
law, Immunome assumes no obligation and does not intend to update
any forward-looking statements included in this press release.
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version on businesswire.com: https://www.businesswire.com/news/home/20241029209009/en/
Immunome Contact: Max Rosett Chief Financial Officer
investors@immunome.com
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